Compile Data Set for Download or QSAR
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Found 369 of affinity data for UniProtKB/TrEMBL: P30547
TargetSubstance-P receptor(GUINEA PIG)
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Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.0590nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
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Curated by PDSP Ki Database
LigandPNGBDBM50000041((+) (2-Methoxy-benzyl)-(2-phenyl-piperidin-3-yl)-a...)
Affinity DataKi:  0.170nMAssay Description:Evaluated for the binding affinity towards NK1 receptor in the striatal membranes of guinea pigMore data for this Ligand-Target Pair
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50000041((+) (2-Methoxy-benzyl)-(2-phenyl-piperidin-3-yl)-a...)
Affinity DataKi:  0.170nMAssay Description:Evaluated for the binding affinity towards NK1 receptor in the striatal membranes of guinea pigMore data for this Ligand-Target Pair
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM86055(SSR240600)
Affinity DataKi:  0.230nMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  0.240nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50116074(CHEMBL66635 | N-[5-(3-Carbamoylmethyl-2-oxo-[1,4']...)
Affinity DataKi:  0.400nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50000040(((2S,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl...)
Affinity DataKi:  0.550nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50116090(1-(2-{1'-[5-[(3,5-Dichloro-benzoyl)-ethyl-amino]-3...)
Affinity DataKi:  0.600nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50116082(3,5-Dichloro-N-(3-(3,4-dichloro-phenyl)-5-{3-[2-(2...)
Affinity DataKi:  0.600nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50116080(3,5-Dichloro-N-{3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  0.700nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50116091(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-5-(3-dimet...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50116087(3,5-Dichloro-N-{3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50116076(CHEMBL441252 | N-[5-(3-Carbamoylmethyl-2-oxo-[1,4'...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50116083(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-5-(3-dimet...)
Affinity DataKi:  0.800nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50116089(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-5-(3-dimet...)
Affinity DataKi:  1nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50366786(CHEMBL540651)
Affinity DataKi:  1nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50116077(3,5-Dichloro-N-{3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  1nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50116088(3,5-Dichloro-N-(3-(3,4-dichloro-phenyl)-5-{3-[2-(2...)
Affinity DataKi:  1.10nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50116075(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  1.20nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50116075(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  1.20nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50116078(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  1.30nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50116085(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  1.5nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50116084(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-methoxyi...)
Affinity DataKi:  2nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50116074(CHEMBL66635 | N-[5-(3-Carbamoylmethyl-2-oxo-[1,4']...)
Affinity DataKi:  2nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50175522(1-{2-[3-((S)-3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  2.12nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM84953(MDL 105,212A (R)-enantiomer)
Affinity DataKi:  2.99nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50116086(3,5-Dichloro-N-(3-(3,4-dichloro-phenyl)-5-{3-[2-(2...)
Affinity DataKi:  3nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50030178((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataKi:  3.13nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50110663(3,5-Dichloro-N-[3-(3,4-dichloro-phenyl)-2-[(Z)-met...)
Affinity DataKi:  5nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50290297(1-{2-[(R)-3-(3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  5.88nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50033658(Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Sarcosine-Leu-Met(...)
Affinity DataKi:  20nMAssay Description:Evaluated for the binding affinity against NK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50029885((3aR,7aR)-2-[1-Imino-2-(2-methoxy-phenyl)-ethyl]-7...)
Affinity DataKi:  36nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataKi:  51nMAssay Description:Evaluated for the binding affinity against NK1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM84954(CAS_6437864 | FK 224 | NSC_6437864)
Affinity DataKi:  98.7nMMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails PubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50175494(1-{2-[(R)-3-(3,4-Dichloro-phenyl)-1-(3,4,5-trimeth...)
Affinity DataKi:  183nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50071112(CHEMBL56835 | N-[4-(4-Acetylamino-4-phenyl-piperid...)
Affinity DataKi:  217nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM82262(ZM253,270)
Affinity DataKi:  9.77E+3nMMore data for this Ligand-Target Pair
In DepthDetails PubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50470591(CHEMBL124208)
Affinity DataKi: <1.00E+4nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 1 from guinea pig tracheaMore data for this Ligand-Target Pair
Ligand InfoPC cidPC sid
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50070546(1-(2-{(S)-3-(3,4-Dichloro-phenyl)-1-[2-(3-isopropo...)
Affinity DataIC50:  0.0190nMAssay Description:Neurokinin (NK1) receptor antagonistic activity was evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50001450((SP)Arg-Pro-Lys-Pro-Gln-Gln-Phe-Phe-Gly-Leu-Met-NH...)
Affinity DataIC50:  0.0700nMAssay Description:Binding affinity towards Tachykinin receptor 1 binding in guinea pig cerebral cortex membranes was determined using [3H]SP as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50070548(1-(2-{3-(3,4-Dichloro-phenyl)-1-[2-(3-isopropoxy-p...)
Affinity DataIC50:  0.310nMAssay Description:Neurokinin (NK1) receptor antagonistic activity was evaluated.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50000040(((2S,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl...)
Affinity DataIC50:  0.400nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1 in guinea pig brain using [125I]-labeled Boltan-Hunter substance P as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50000040(((2S,3S)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl...)
Affinity DataIC50:  0.560nMAssay Description:Antagonism of the guinea pig tachykinin NK1 receptorMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50049338(CHEMBL353093 | N-[1-{[Acetyl-(2-methoxy-benzyl)-am...)
Affinity DataIC50:  0.880nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1 in guinea pig brain using [125I]-labeled Boltan-Hunter substance P as radioligandMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50066238((S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(b...)
Affinity DataIC50:  1nMAssay Description:Tachykinin receptor 1 agonistic activity as inhibition of contractions evoked by 4 nM [Sar9,Met(O2)11]-SP in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50030174((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  1.10nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50280461(((2R,3R)-2-Benzhydryl-1-aza-bicyclo[2.2.2]oct-3-yl...)
Affinity DataIC50:  1.20nMAssay Description:Binding affinity towards Tachykinin receptor 1 binding in guinea pig cerebral cortex membranes was determined using [3H]SP as the radioligandMore data for this Ligand-Target Pair
In DepthDetails Article
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50066193((S)-Pyrrolidine-1,2-dicarboxylic acid 2-{[(S)-1-(b...)
Affinity DataIC50:  1.20nMAssay Description:Tachykinin receptor 1 agonistic activity as inhibition of contractions evoked by 4 nM [Sar9,Met(O2)11]-SP in guinea pig ileumMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50030199((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  1.70nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSubstance-P receptor(GUINEA PIG)
Sanofi-SynthÉLabo Recherche

Curated by PDSP Ki Database
LigandPNGBDBM50030178((R)-4-Hydroxy-1-(1-methyl-1H-indole-3-carbonyl)-py...)
Affinity DataIC50:  1.70nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
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