Affinity DataKi: 0.170nMAssay Description:Evaluated for the binding affinity towards NK1 receptor in the striatal membranes of guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.170nMAssay Description:Evaluated for the binding affinity towards NK1 receptor in the striatal membranes of guinea pigMore data for this Ligand-Target Pair
Affinity DataKi: 0.400nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 0.600nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 0.700nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 0.800nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 1nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 1.10nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 1.20nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 1.30nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 1.5nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 2nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 3nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 5nMAssay Description:In vitro binding to Tachykinin receptor 1More data for this Ligand-Target Pair
Affinity DataKi: 20nMAssay Description:Evaluated for the binding affinity against NK1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: 51nMAssay Description:Evaluated for the binding affinity against NK1 receptorMore data for this Ligand-Target Pair
Affinity DataKi: <1.00E+4nMAssay Description:The compound was tested for binding affinity against Tachykinin receptor 1 from guinea pig tracheaMore data for this Ligand-Target Pair
Affinity DataIC50: 0.0190nMAssay Description:Neurokinin (NK1) receptor antagonistic activity was evaluated.More data for this Ligand-Target Pair
Affinity DataIC50: 0.0700nMAssay Description:Binding affinity towards Tachykinin receptor 1 binding in guinea pig cerebral cortex membranes was determined using [3H]SP as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.310nMAssay Description:Neurokinin (NK1) receptor antagonistic activity was evaluated.More data for this Ligand-Target Pair
Affinity DataIC50: 0.400nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1 in guinea pig brain using [125I]-labeled Boltan-Hunter substance P as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 0.560nMAssay Description:Antagonism of the guinea pig tachykinin NK1 receptorMore data for this Ligand-Target Pair
Affinity DataIC50: 0.880nMAssay Description:Inhibitory activity of the compound against Tachykinin receptor 1 in guinea pig brain using [125I]-labeled Boltan-Hunter substance P as radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1nMAssay Description:Tachykinin receptor 1 agonistic activity as inhibition of contractions evoked by 4 nM [Sar9,Met(O2)11]-SP in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 1.10nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Binding affinity towards Tachykinin receptor 1 binding in guinea pig cerebral cortex membranes was determined using [3H]SP as the radioligandMore data for this Ligand-Target Pair
Affinity DataIC50: 1.20nMAssay Description:Tachykinin receptor 1 agonistic activity as inhibition of contractions evoked by 4 nM [Sar9,Met(O2)11]-SP in guinea pig ileumMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair
Affinity DataIC50: 1.70nMAssay Description:In vitro binding affinity against substance P receptor using [3H]SP as radioligand in guinea pig lung membraneMore data for this Ligand-Target Pair